Candesartan exhibits low intrinsic permeation capacity and affects buccal tissue viability and integrity: An ex vivo study in porcine buccal mucosa
Candesartan is a nonpeptide angiotensin II receptor blocker that selectively binds to angiotensin II receptor subtype 1. It is administered orally in its ester form (candesartan cilexetil). However, its poor aqueous solubility results in its low bioavailability; therefore, other routes of administra...
- Autores:
-
Garcia-Tarazona, Yenny M.
Morantes, Sandra Johanna
Gordillo, José Francisco Ibla
Sepúlveda, Paula
Ramos, Freddy A.
Lafaurie, Gloria Inés
- Tipo de recurso:
- Article of journal
- Fecha de publicación:
- 2023
- Institución:
- Universidad El Bosque
- Repositorio:
- Repositorio U. El Bosque
- Idioma:
- eng
- OAI Identifier:
- oai:repositorio.unbosque.edu.co:20.500.12495/11246
- Acceso en línea:
- http://hdl.handle.net/20.500.12495/11246
https://doi.org/10.1016/j.ejps.2023.106495
- Palabra clave:
- Permeabilidad bucal
Candesartán
Histología Índice TR
Ensayo MTT
Buccal permeability
Candesartan
Histology TR index
MTT assay
- Rights
- openAccess
- License
- Atribución 4.0 Internacional